Towards broadspectrum antiprotozoal agents

by Kelly Chibale
Published 2003-01-01

Cell-Based Medicinal Chemistry Optimization of High Throughput Screening Hits towards Orally Active Antimalarial and Antituberculosis Agents

by Kelly Chibale
Published 2017-12-01

Introduction to the 1st Molecules Medicinal Chemistry Symposium (MMCS), Barcelona, 8 September 2017

by Diego Muñoz-Torrero, Kelly Chibale
Published 2017-12-01

Novel tetracyclic structures from the synthesis of thiolactone-isatin hybrids

by Renate Hazel Hans, Hong Su, Kelly Chibale
Published 2010-07-01

Synthesis and In Vitro Antiprotozoan Evaluation of 4-/8-Aminoquinoline-based Lactams and Tetrazoles

by Matshawandile Tukulula, Stefan Louw, Mathew Njoroge, Kelly Chibale
Published 2020-12-01

The Role of Natural Products in Drug Discovery and Development against Neglected Tropical Diseases

by Peter Mubanga Cheuka, Godfrey Mayoka, Peggoty Mutai, Kelly Chibale
Published 2016-12-01

Inhibition of trypanothione reductase and glutathione reductase by ferrocenic 4-aminoquinoline ureas

by Margaret A.L. Blackie, Ahilan Saravanamuthu, Alan H. Fairlamb, Kelly Chibale
Published 2008-03-01

Synthesis of novel β-lactams and in vitro evaluation against the human malaria parasite Plasmodium falciparum

by Margaret A.L. Blackie, Tzu-Shean Feng, Peter J Smith, Kelly Chibale
Published 2016-03-01

Intestinal Transport Characteristics and Metabolism of C-Glucosyl Dihydrochalcone, Aspalathin

by Sandra Bowles, Elizabeth Joubert, Dalene de Beer, Johan Louw, Christel Brunschwig, Mathew Njoroge, Nina Lawrence, Lubbe Wiesner, Kelly Chibale, Christo Muller
Published 2017-03-01

Synthesis of 2-amino-3-arylpropan-1-ols and 1-(2,3-diaminopropyl)-1,2,3-triazoles and evaluation of their antimalarial activity

by Matthias D’hooghe, Stéphanie Vandekerckhove, Karen Mollet, Karel Vervisch, Stijn Dekeukeleire, Liesbeth Lehoucq, Carmen Lategan, Peter J. Smith, Kelly Chibale, Norbert De Kimpe
Published 2011-12-01

Anticancer properties of distinct antimalarial drug classes.

by Rob Hooft van Huijsduijnen, R Kiplin Guy, Kelly Chibale, Richard K Haynes, Ingmar Peitz, Gerhard Kelter, Margaret A Phillips, Jonathan L Vennerstrom, Yongyuth Yuthavong, Timothy N C Wells
Published 2013-01-01

Potentiation of rifampin activity in a mouse model of tuberculosis by activation of host transcription factor EB.

by Ruslana Bryk, Shashirekha Mundhra, Xiuju Jiang, Madeleine Wood, Daniel Pfau, Elaina Weber, Suna Park, Li Zhang, Colin Wilson, Renier Van der Westhuyzen, Leslie Street, Kelly Chibale, Matthew Zimmerman, Véronique Dartois, Nunzia Pastore, Andrea Ballabio, Natalie Hawryluk, Stacie Canan, Vikram Khetani, Joseph Camardo, Carl Nathan
Published 2020-06-01

The Next Generation Scientist program: capacity-building for future scientific leaders in low- and middle-income countries

by Goonaseelan Pillai, Kelly Chibale, Edwin C. Constable, Akiko N. Keller, Marcelo M. Gutierrez, Fareed Mirza, Christian Sengstag, Collen Masimirembwa, Paolo Denti, Gary Maartens, Michèle Ramsay, Bernhards Ogutu, Eyasu Makonnen, Richard Gordon, Carlos Gil Ferreira, Fernando Alberto Goldbaum, Wim M. S. Degrave, Jonathan Spector, Brigitta Tadmor, Hedwig J. Kaiser
Published 2018-10-01

Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box

by Janette Reader, Mariëtte E. van der Watt, Dale Taylor, Claire Le Manach, Nimisha Mittal, Sabine Ottilie, Anjo Theron, Phanankosi Moyo, Erica Erlank, Luisa Nardini, Nelius Venter, Sonja Lauterbach, Belinda Bezuidenhout, Andre Horatscheck, Ashleigh van Heerden, Natalie J. Spillman, Anne N. Cowell, Jessica Connacher, Daniel Opperman, Lindsey M. Orchard, Manuel Llinás, Eva S. Istvan, Daniel E. Goldberg, Grant A. Boyle, David Calvo, Dalu Mancama, Theresa L. Coetzer, Elizabeth A. Winzeler, James Duffy, Lizette L. Koekemoer, Gregory Basarab, Kelly Chibale, Lyn-Marié Birkholtz
Published 2021-01-01