Synergistic catalysis: highly diastereoselective benzoxazole addition to Morita-Baylis-Hillman carbonates
An expedited method has been developed for the diastereoselective synthesis of highly functionalized alkyl-azaarene systems with good yields and high diastereoselectivities (>15 : 1 dr). The methodology includes a synergistic catalysis event involving organometallic (10 mol% AgOAc) activation of...
| Main Authors: | , , , , , , |
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| Format: | Article |
| Language: | English |
| Published: |
2014-05-20.
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| Subjects: | |
| Online Access: | Get fulltext |