Novel, potent antagonists of capsaicin
The aim of this project was to explore and refine the conformational rationale for the activity of capsazepine (CPZ) as a blocker of the ion channel TRPV1 (transient receptor potential vanilloid type 1), by the synthesis and biological evaluation of further conformational constrained capsaicin analo...
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University College London (University of London)
2005
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Online Access: | http://ethos.bl.uk/OrderDetails.do?uin=uk.bl.ethos.684729 |