Triazolobenzodiazepines and -triazepines as protein interaction inhibitors targeting bromodomains of the BET family

Benzodiazepines are psychoactive drugs with anxiolytic, sedative, skeletal muscle relaxant and amnestic properties. Recently triazolobenzodiazepines have been also described as potent and highly selective protein interaction inhibitors of bromodomain and extra-terminal (BET) proteins, a family of tr...

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Bibliographic Details
Main Author: Wrobel, Matthias
Format: Others
Published: Ludwig-Maximilians-Universität München 2014
Subjects:
Online Access:http://edoc.ub.uni-muenchen.de/16562/1/Wrobel_Matthias_A.pdf
http://nbn-resolving.de/urn:nbn:de:bvb:19-165623