Click Conjugation of Boron Dipyrromethene (BODIPY) Fluorophores to EGFR-Targeting Linear and Cyclic Peptides

Through a simple 1,3-cycloaddition reaction, three BODIPY-peptide conjugates that target the extracellular domain of the epidermal growth factor receptor (EGFR) were prepared and their ability for binding to EGFR was investigated. The peptide ligands K(N<sub>3</sub>)LARLLT and its cyclic...

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Bibliographic Details
Main Authors: Tyrslai M. Williams, Nichole E. M. Kaufman, Zehua Zhou, Sitanshu S. Singh, Seetharama D. Jois, Maria da Graça H. Vicente
Format: Article
Language:English
Published: MDPI AG 2021-01-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/26/3/593