One-Pot Synthesis of Novel 2,3-Dihydro-1H-indazoles

A copper(I)-mediated one-pot synthesis of 2,3-dihydro-1H-indazole heterocycles has been developed. This synthetic route provides the desired indazoles in moderate to good yields (55%–72%) which are substantially better than those achievable with an alternative two-step reaction sequence. The reactio...

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Bibliographic Details
Main Authors: Antonio J. Lepore, Gary W. Breton
Format: Article
Language:English
Published: MDPI AG 2011-11-01
Series:Molecules
Subjects:
Online Access:http://www.mdpi.com/1420-3049/16/11/9553/