Preparation of E-1,3-diaminoethenyl functional groups by the reaction of enol tosylate of alpha-formylglycine with primary and secondary amines
The E-1,3-diaminoethenyl functional group is a potentially useful synthon. A number of examples of E-1,3-diaminoethenyl functional groups were prepared in good yield starting from an E-enol tosylate of a serine based diketopiperazine and 1°- or 2° amine nucleophiles. The reaction proceeds via a ster...
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| Format: | Article |
| Language: | English |
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Growing Science
2016-03-01
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| Series: | Current Chemistry Letters |
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| Online Access: | http://www.growingscience.com/ccl/Vol5/ccl_2016_1.pdf |