Dynamics and ligand-induced conformational changes in human prolyl oligopeptidase analyzed by hydrogen/deuterium exchange mass spectrometry

by Alexandra Tsirigotaki, Roos Van Elzen, Pieter Van Der Veken, Anne-Marie Lambeir, Anastassios Economou
Published 2017-05-01

Molecular Imaging of Apoptosis: The Case of Caspase-3 Radiotracers

by Lucas Beroske, Tim Van den Wyngaert, Sigrid Stroobants, Pieter Van der Veken, Filipe Elvas
Published 2021-04-01

Asymmetric synthesis of γ-chloro-α,β-diamino- and β,γ-aziridino-α-aminoacylpyrrolidines and -piperidines via stereoselective Mannich-type additions of N-(diphenylmethylene)glycinam...

by Gert Callebaut, Sven Mangelinckx, Pieter Van der Veken, Karl W. Törnroos, Koen Augustyns, Norbert De Kimpe
Published 2012-12-01

An essential signal peptide peptidase identified in an RNAi screen of serine peptidases of Trypanosoma brucei.

by Catherine X Moss, Elaine Brown, Alana Hamilton, Pieter Van der Veken, Koen Augustyns, Jeremy C Mottram
Published 2015-01-01

ClpP Protease, a Promising Antimicrobial Target

by Carlos Moreno-Cinos, Kenneth Goossens, Irene G. Salado, Pieter Van Der Veken, Hans De Winter, Koen Augustyns
Published 2019-05-01

Circulating Stromal Cell-Derived Factor 1α Levels in Heart Failure: A Matter of Proper Sampling.

by Lesley Baerts, Yannick Waumans, Inger Brandt, Wolfgang Jungraithmayr, Pieter Van der Veken, Marc Vanderheyden, Ingrid De Meester
Published 2015-01-01

Prolyl Carboxypeptidase Mediates the C-Terminal Cleavage of (Pyr)-Apelin-13 in Human Umbilical Vein and Aortic Endothelial Cells

by Emilie De Hert, An Bracke, Isabel Pintelon, Eline Janssens, Anne-Marie Lambeir, Pieter Van Der Veken, Ingrid De Meester
Published 2021-06-01

The effect of pharmacological inhibition of Serine Proteases on neuronal networks in vitro

by Sebastiaan Van De Vijver, Stephan Missault, Jeroen Van Soom, Pieter Van Der Veken, Koen Augustyns, Jurgen Joossens, Stefanie Dedeurwaerdere, Michele Giugliano
Published 2019-04-01

In Vitro Evaluation of the Squaramide-Conjugated Fibroblast Activation Protein Inhibitor-Based Agents AAZTA⁵.SA.FAPi and DOTA.SA.FAPi

by Euy Sung Moon, Yentl Van Rymenant, Sandeep Battan, Joni De Loose, An Bracke, Pieter Van der Veken, Ingrid De Meester, Frank Rösch
Published 2021-06-01

Selective Activity-Based Probes Targeting Fibroblast Activation Protein (FAP)

by Johannes Vrijdag, Anvesh Jallapally, An De Decker, Koen Janssen, Filipe Elvas, Steven Staelens, Ingrid De Meester, Koen Augustyns, Anne-Marie Lambeir, Pieter Van der Veken
Published 2019-08-01

In Vitro and In Situ Activity-Based Labeling of Fibroblast Activation Protein with UAMC1110-Derived Probes

by Yentl Van Rymenant, Muhammet Tanc, Roos Van Elzen, An Bracke, Olivier De Wever, Koen Augustyns, Anne-Marie Lambeir, Mark Kockx, Ingrid De Meester, Pieter Van Der Veken
Published 2021-04-01

The Effect of a Novel Serine Protease Inhibitor on Inflammation and Intestinal Permeability in a Murine Colitis Transfer Model

by Hanne Van Spaendonk, Hanne Van Spaendonk, Hannah Ceuleers, Hannah Ceuleers, Annemieke Smet, Annemieke Smet, Maya Berg, Jurgen Joossens, Pieter Van der Veken, Pieter Van der Veken, Sven M. Francque, Sven M. Francque, Sven M. Francque, Anne-Marie Lambeir, Anne-Marie Lambeir, Joris G. De Man, Joris G. De Man, Ingrid De Meester, Ingrid De Meester, Koen Augustyns, Koen Augustyns, Benedicte Y. De Winter, Benedicte Y. De Winter, Benedicte Y. De Winter
Published 2021-06-01

Blockade of fibroblast activation protein in combination with radiation treatment in murine models of pancreatic adenocarcinoma.

by Andrew J Gunderson, Tomoko Yamazaki, Kayla McCarty, Michaela Phillips, Alejandro Alice, Shelly Bambina, Lauren Zebertavage, David Friedman, Benjamin Cottam, Pippa Newell, Michael J Gough, Marka R Crittenden, Pieter Van der Veken, Kristina H Young
Published 2019-01-01

Targeting fibroblast activation protein (FAP): next generation PET radiotracers using squaramide coupled bifunctional DOTA and DATA5m chelators

by Euy Sung Moon, Filipe Elvas, Gwendolyn Vliegen, Stef De Lombaerde, Christel Vangestel, Sven De Bruycker, An Bracke, Elisabeth Eppard, Lukas Greifenstein, Benedikt Klasen, Vasko Kramer, Steven Staelens, Ingrid De Meester, Pieter Van der Veken, Frank Rösch
Published 2020-07-01

Selective Glucocorticoid Receptor Properties of GSK866 Analogs with Cysteine Reactive Warheads

by Chandra S. Chirumamilla, Ajay Palagani, Balu Kamaraj, Ken Declerck, Marinus W. C. Verbeek, Ryabtsova Oksana, Karolien De Bosscher, Nadia Bougarne, Bart Ruttens, Kris Gevaert, René Houtman, Winnok H. De Vos, Jurgen Joossens, Pieter Van Der Veken, Koen Augustyns, Xaveer Van Ostade, Annemie Bogaerts, Hans De Winter, Wim Vanden Berghe
Published 2017-11-01