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241“... nuclear warhead attached to the missile in 1966. Since then, China has become one of the countries...”
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242by Patel, Neki Vijay“...' was exploited to incorporate the HA 'warhead'. This 'small molecule-peptide chimera library' enabled...”
Published 2012
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243by Sivels, Ciara (Ciara Brooke)“.... Speculations are that this test was conducted to further develop a warhead small enough to fit...”
Published 2013
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244“... is one of the key issues to assess the damage efficiency of the warhead. However, limited work has been...”
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245“...; an “anchor” to bind to an E3 ubiquitin ligase and a “warhead” to bind to a protein of interest, connected...”
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246by Wen-Hao Guo, Xiaoli Qi, Xin Yu, Yang Liu, Chan-I Chung, Fang Bai, Xingcheng Lin, Dong Lu, Lingfei Wang, Jianwei Chen, Lynn Hsiao Su, Krystle J. Nomie, Feng Li, Meng C. Wang, Xiaokun Shu, José N. Onuchic, Jennifer A. Woyach, Michael L. Wang, Jin Wang“.... Here, the authors show that reversible covalent warhead chemistry improves PROTAC intracellular...”
Published 2020-08-01
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248by Mladenovic, Milena“... of the electrophilic warhead of the inhibitor (both substitituted and not) and molecular moieties simulating a very...”
Published 2008
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Doctoral Thesis -
249by Mark G. Anderson, Qian Zhang, Luis E. Rodriguez, Claudie M. Hecquet, Cherrie K. Donawho, Peter J. Ansell, Edward B. Reilly“... pyrrolobenzodiazepine (PBD) dimer cytotoxin, an emerging class of warheads with enhanced potency and broader anticancer...”
Published 2021-06-01
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250by Eun Lee, Hyewon Cho, Da Kyung Lee, JuHyun Ha, Byeong Jo Choi, Ji Hye Jeong, Jae-Ha Ryu, Jong Soon Kang, Raok Jeon“... conformation and introduced an electrophilic warhead for targeting Cys481. In this article, we have described...”
Published 2020-10-01
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251by Alexander, Nathan Austin“... which incorporate an azobenzene photoswitch, a peptidyl backbone and a trifluoromethyl ketone warhead...”
Published 2008
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252“... that the warhead modification of these CTSS inhibitor analogs increased inhibitory ability such that an IC50 value...”
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253“... United States Forces Korea and the problem of nuclear development and warhead launch. If these problems...”
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254by Akhil, G“... are crucial for a greater warhead effectiveness, and minimizing the interception time is important...”
Published 2018
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255by Aziz, Shaista“... inhibitors of K-RasG12C incorporating the cyclohexadienone moiety as the thiol-reactive warhead to covalently...”
Published 2017
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256“..., the power of shrapnel and manufacturing cost, the 8-prism are better choices for cluster warhead underwater...”
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257“...-bullets capable of holding both an anticancer drug and DNA cleaving warhead with an oligonucleotide on a...”
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258by Miller, Zachary C.“... inhibitors rely on the combination a peptide backbone and reactive electrophilic warhead to target...”
Published 2018
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259by Zerfas, Breanna L.“... work towards establishing a novel cyclic peptide library incorporating a 2-APBA warhead...”
Published 2017
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260by Hyewon Cho, Eun Lee, Hye Ah Kwon, Lee Seul, Hui-Jeon Jeon, Ji Hoon Yu, Jae-Ha Ryu, Raok Jeon“... the modification of pyranochromenone at the C7 position. Pyranochromenone compounds with an electrophilic warhead...”
Published 2020-10-01
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