The design, synthesis and protease inhibitor properties of latent reactive amino acid analogues

The design, synthesis and protease inhibitor properties of latent reactive amino acid analogues

This thesis examines the synthesis and proteolytic properties of a new class of latent reactive amino acid analogue, eg: 1-(N-Phthaloyl-Lphenylalanyl)-2-hydroxymethylpyrrole 2.52, designed to inhibit serine proteases and the HN protease. Chapter One discusses the possible mode of protease inhibitio...

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Bibliographic Details
Main Author:	Litten, J. Christopher
Language:	en
Published:	University of Canterbury. Chemistry 2012
Online Access:	http://hdl.handle.net/10092/7300

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