Synthesis of 3-arylisoxazoles and 5-arylisoxazoles

Synthesis of 3-arylisoxazoles and 5-arylisoxazoles

The goal of this research project was to synthesize a small library of 3- and 5-arylisoxazoles. These compounds are of interest because of potential biological activity similar to Fipronil. Fipronil is used commercially in the agrochemical industry and exhibits pesticidal activity as a noncompetitiv...

Full description

Bibliographic Details
Main Author:	Pertler, Stephanie L.
Other Authors:	Sammelson, Robert E.
Format:	Others
Published:	2011
Subjects:	Oxazoles > Synthesis. GABA > Inhibitors > Synthesis.
Online Access:	http://cardinalscholar.bsu.edu/handle/handle/188154 http://liblink.bsu.edu/uhtbin/catkey/1348869

Similar Items

Design, synthesis and biological evaluation of 3-(2-aminooxazol-5-yl)-2H-chromen-2-one derivatives
by: Saloni Kakkar, et al.
Published: (2018-12-01)

Design, synthesis and biological evaluation of 3-(2-aminooxazol-5-yl)-2H-chromen-2-one derivatives
by: Kakkar, S., et al.
Published: (2018)

Development of a method for the synthesis of 2,4,5-trisubstituted oxazoles composed of carboxylic acid, amino acid, and boronic acid
by: Kohei Yamada, et al.
Published: (2017-07-01)

Design, synthesis and biological evaluation of 3-(2-aminooxazol-5-yl)-2H-chromen-2-one derivatives
by: Kakkar, S, et al.
Published: (2018)

Synthesis and Herbicidal Activities of Novel 4-(4-(5-methyl-3-arylisoxazol-4-yl)thiazol-2-yl)piperidyl Carboxamides and Thiocarboxamides
by: Ai-Dong Zhang, et al.
Published: (2009-03-01)

Recent Advances in the Synthesis of Oxazole-Based Molecules via van Leusen Oxazole Synthesis
by: Xunan Zheng, et al.
Published: (2020-03-01)

Design, synthesis and biological potential of heterocyclic benzoxazole scaffolds as promising antimicrobial and anticancer agents
by: Kakkar, S, et al.
Published: (2018)

Design, synthesis and cholinesterase inhibitory properties of new oxazole benzylamine derivatives
by: Ivana Šagud, et al.
Published: (2020-01-01)

Synthesis of 4-alkyl-3,5-diamino-1-phenylpyrazoles
by: Dunham, Jason C.
Published: (2011)

Total Synthesis of Bacterial 5-(3-Indolyl)oxazole Alkaloids: Pimprinols A–C
by: Tímea Szabó, et al.
Published: (2019-10-01)

Synthesis of Highly Substituted Oxazoles through Iodine(III)-Mediated Reactions of Ketones with Nitriles
by: Yuji Hanzawa, et al.
Published: (2012-09-01)

Synthesis and biological evaluation of (3-arylisoxazol-5-yl) methyl 6-fluoro-4-oxo-4H-chromene-2-carboxylates as antioxidant and antimicrobial agents
by: Battula Kumaraswamy, et al.
Published: (2017-01-01)

Studies Toward the Total Synthesis and Structure Determination of Leiodelide A
by: Chellat, Mathieu François
Published: (2011)

Solid Phase versus Solution Phase Synthesis of Heterocyclic Macrocycles
by: Shelli R. McAlpine, et al.
Published: (2013-01-01)

Design, synthesis, molecular docking and anticonvulsant evaluation of 6-methyl-2-arylaminopyrimidin-4(3H)-one
by: Hanna Severina, et al.
Published: (2020-04-01)

Synthetic utility of 5-amino-6-cyano-2-phenylthieno[2,3-d] oxazole
by: Kanetkar V.R., et al.
Published: (2005-01-01)

Thiazole and Oxazole Alkaloids: Isolation and Synthesis
by: Gloria Serra, et al.
Published: (2010-11-01)

Antiplasmodial dihetarylthioethers target the coenzyme A synthesis pathway in Plasmodium falciparum erythrocytic stages
by: Thomas Weidner, et al.
Published: (2017-05-01)

Synthetic utility of 5-amino-6-cyano-2-phenylthieno[2,3-d] oxazole
by: V. R. KANETKAR, et al.
Published: (2005-11-01)

1,3-Oxazol-4-ylphosphonium salts as new non-peptide inhibitors of furin
by: T. V. Osadchuk, et al.
Published: (2019-08-01)

Synthesis and Bioactivity of N-Benzoyl-N'-[5-(2'-substituted phenyl)-2-furoyl] Semicarbazide Derivatives
by: Zining Cui, et al.
Published: (2010-06-01)

Macrooxazoles A–D, New 2,5-Disubstituted Oxazole-4-Carboxylic Acid Derivatives from the Plant Pathogenic Fungus <i>Phoma macrostoma</i>
by: Blondelle Matio Kemkuignou, et al.
Published: (2020-11-01)

Topics In Synthetic Methodology : From Heterocycles To Hydride Transfers
by: Srimannarayana, Malempati
Published: (2013)

Synthesis of new derivatives of 3-azabicyclo[3.3.1]nonan based on N-(2-hydroxy-3,5-dinitrophenyl)benzamide
by: Loik Mukhtorov, et al.
Published: (2021-01-01)

Development of Novel Methodologies for the Synthesis and Functionalization of Nitrogen Heterocycles
by: Counceller, Carla Marie
Published: (2010)

Isomerization of 5-(2<i>H</i>-Azirin-2-yl)oxazoles: An Atom-Economic Approach to 4<i>H</i>-Pyrrolo[2,3-<i>d</i>]oxazoles
by: Timur O. Zanakhov, et al.
Published: (2021-03-01)

Discontinuous DNA synthesis in mammalian cells.
by: Horwitz, Henry Bennet
Published: (2008)

Synthesis, characterization and comparative study the microbial activity of some heterocyclic compounds containing oxazole and benzothiazole moieties
by: Ivan H.R. Tomi, et al.
Published: (2015-07-01)

A modified approach for the synthesis of biologically relevant 5-substituted-2-N-aryl-1,3-oxazole derivatives in mild conditions
by: R. Udhayasurian, et al.
Published: (2020-01-01)

Cyclization of Activated Methylene Isocyanides with Methyl N(N),N′-Di(tri)substituted Carbamimidothioate: A Novel Entry for the Synthesis of N,1-Aryl-4-tosyl/ethoxycarbonyl-1H-imidazol-5-amines
by: Dukanya Dukanya, et al.
Published: (2019-07-01)

Expedient synthesis of chiral poly-substituted morpholine and oxazepine derivatives for the preparation of cyclophilin A inhibitors
by: Bilbeisi, Rana A., 1983-
Published: (2008)

The synthesis of 3,5-disubstituted indolizidines
by: Cheesman, Penelope, Sue
Published: (2017)

Synthesis of modified small peptide inhibitors
by: Norman, S. E.
Published: (1988)

Synthesis of 1,4-imino-L-lyxitols modified at C-5 and their evaluation as inhibitors of GH38 α-mannosidases
by: Maroš Bella, et al.
Published: (2018-08-01)

Solvothermal Synthesis of Multiple Dihydropyrimidinones at a Time as Inhibitors of Eg5
by: Xiao-Qiang Jiang, et al.
Published: (2021-03-01)

Synthesis and characterization of some heterocyclic including oxazoles,Thiazoles, Pyridazines, phthalizines and Pyrazoles with evaluating of biological activity.
by: Baghdad Science Journal
Published: (2013-09-01)

Total Synthesis of Phorbazole B
by: Yngve Guttormsen, et al.
Published: (2020-10-01)

Design and Synthesis of New Benzo[d]oxazole-Based Derivatives and Their Neuroprotective Effects on β-Amyloid-Induced PC12 Cells
by: Zheng Liu, et al.
Published: (2020-11-01)

Synthesis of 6-guanidinobenzoxazinones as potential inhibitors of trypsin-like enzymes
by: Silveira, Alvito J.
Published: (2009)

Synthesis and PI 3-Kinase Inhibition Activity of Some Novel 2,4,6-Trisubstituted 1,3,5-Triazines
by: Ronald A. Nelson, et al.
Published: (2018-07-01)