Truncated azinomycin analogues intercalate into DNA.
No === The design and synthesis of a potentially more therapeutically-viable azinomycin analogue 4 based upon 3 has been completed. It involved coupling of a piperidine mustard to the acid chloride of the azinomycin chromophore. Both the designed azinomycin analogue 4 and the natural product 3 bind...
Main Authors: | Casely-Hayford, M.A., Pors, Klaus, Patterson, Laurence H., Gerner, C., Neidle, S., Searcey, M. |
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Language: | en |
Published: |
2009
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Subjects: | |
Online Access: | http://hdl.handle.net/10454/3908 |
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