HFIP-Promoted Bischler Indole Synthesis under Microwave Irradiation
1,1,1,3,3,3-Hexafluoropropan-2-ol (HFIP) was found to be effective for the Bischler indole synthesis under microwave irradiation in the absence of a metal catalyst. Under the catalysis of HFIP, a wide range of α-amino arylacetones were successfully transformed into indole derivatives with m...
Main Authors: | Guangkai Yao, Zhi-Xiang Zhang, Cheng-Bei Zhang, Han-Hong Xu, Ri-Yuan Tang |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2018-12-01
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Series: | Molecules |
Subjects: | |
Online Access: | https://www.mdpi.com/1420-3049/23/12/3317 |
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