Thiazolidin-4-one, azetidin-2-one and 1,3,4-oxadiazole derivatives of isonicotinic acid hydrazide: synthesis and their biological evaluation

Thiazolidin-4-one, azetidin-2-one and 1,3,4-oxadiazole derivatives of isonicotinic acid hydrazide: synthesis and their biological evaluation

A series of thiazolidin-4-one (2a–h; 3a–h), azetidin-2-one (4a–h) and 1,3,4-oxadiazole (5a–h) derivatives of isoninicotinic acid hydrazide (INH) were synthesized in order to obtain new compounds with potential anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation activities. The structur...

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Bibliographic Details
Main Authors:	VIJENDER SINGH, ALKA ARORA, OZAIR ALAM, SUROOR A. KHAN, SADAF J. GILANI
Format:	Article
Language:	English
Published:	Serbian Chemical Society 2011-08-01
Series:	Journal of the Serbian Chemical Society
Subjects:	anti-inflammatory activity analgesic activity ulcerogenic activity lipid peroxidation.
Online Access:	http://www.shd.org.rs/JSCS/Vol76/No8/01_4608_4184.pdf

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