Tetrahydro-iso-alpha Acids Antagonize Estrogen Receptor Alpha Activity in MCF-7 Breast Cancer Cells

Tetrahydro-iso-alpha Acids Antagonize Estrogen Receptor Alpha Activity in MCF-7 Breast Cancer Cells

Tetrahydro-iso-alpha acids commonly called THIAA or Tetra are modified hop acids extracted from hop (Humulus lupulus L.) which are frequently used in brewing industry mainly in order to provide beer bitterness and foam stability. Interestingly, molecular structure of tetrahydro-iso-alpha acids is cl...

Full description

Bibliographic Details
Main Authors:	Maëlle Lempereur, Claire Majewska, Amandine Brunquers, Sumalee Wongpramud, Bénédicte Valet, Philippe Janssens, Monique Dillemans, Laurence Van Nedervelde, Dominique Gallo
Format:	Article
Language:	English
Published:	Hindawi Limited 2016-01-01
Series:	International Journal of Endocrinology
Online Access:	http://dx.doi.org/10.1155/2016/9747863

Similar Items

Inhibition of ISO- Induced Cardiomyoblast Hypertrophy By Estrogen And Estrogen Receptor-alpha Is Protein Phosphatase 1- Dependent
by: Chia-Chien, et al.
Published: (2006)

Tetrahydro iso-alpha acids from hops improve glucose homeostasis and reduce body weight gain and metabolic endotoxemia in high-fat diet-fed mice.
by: Amandine Everard, et al.
Published: (2012-01-01)

Role of estrogen receptor alpha (ER alpha) insulin-like growth factor (IGF)-I-induced responses in MCF-7 breast cancer cells
by: Zhang, Shu
Published: (2010)

Comparative activation of estrogen receptor alpha (er alpha) by endocrine disruptors
by: Wu, Fei
Published: (2010)

Measuring the binding kinetics of estrogen receptor alpha and dietary estrogens
by: Lee, Isaish Chi Kin
Published: (2014)

Autocrine regulation of cell proliferation by estrogen receptor-alpha in estrogen receptor-alpha-positive breast cancer cell lines
by: Pan Zhongzong, et al.
Published: (2009-01-01)

Dual targeting of estrogen receptor α and estrogen-related receptor α: a novel endocrine therapy for endometrial cancer
by: Mao X, et al.
Published: (2019-08-01)

ANTIPROLIFERATIVE ACTIVITY OF RECOMBINANT HUMAN INTERFERON ALPHA2B ON ESTROGEN POSITIVE HUMAN BREAST CANCER MCF-7 CELL LINE
by: Ratih Asmana Ningrum, et al.
Published: (2015-05-01)

Characterization of a novel small molecule subtype specific estrogen-related receptor alpha antagonist in MCF-7 breast cancer cells.
by: Michael J Chisamore, et al.
Published: (2009-05-01)

Circadian modulation of the estrogen receptor alpha transcription
by: Villa, Linda Monique
Published: (2017)

Expression of Estrogen Receptor Alpha in Malignant Melanoma
by: Parvin Rajabi, et al.
Published: (2017-01-01)

Estrogen receptor alpha localization in the testes of men with normal spermatogenesis Estrogen receptor alpha localization in the testes of men with normal spermatogenesis
by: Eliza Filipiak, et al.
Published: (2012-10-01)

Investigation of the cellular and physiological effects of 5 alpha-tetrahydro reduced glucocorticoids in vitro and in vivo
by: Yang, Chenjing
Published: (2010)

17β-Estradiol and/or estrogen receptor alpha signaling blocks protein phosphatase 1 mediated ISO induced cardiac hypertrophy.
by: Hsin-Yuan Fang, et al.
Published: (2018-01-01)

Estrogen signalling and the metabolic syndrome: targeting the hepatic estrogen receptor alpha action.
by: Marko Matic, et al.
Published: (2013-01-01)

Estrogen/estrogen receptor alpha signaling in mouse posterofrontal cranial suture fusion.
by: Aaron W James, et al.
Published: (2009-09-01)

Computer-Aided Ligand Discovery for Estrogen Receptor Alpha
by: Divya Bafna, et al.
Published: (2020-06-01)

Estrogen Receptors Alpha and Beta in Acute Myeloid Leukemia
by: Alessia Roma, et al.
Published: (2020-04-01)

Activation of estrogen receptor alpha induces beiging of adipocytes
by: Roberta S. Santos, et al.
Published: (2018-12-01)

Estrogen receptor alpha and nuclear factor Y coordinately regulate the transcription of the SUMO-conjugating UBC9 gene in MCF-7 breast cancer cells.
by: Shibo Ying, et al.
Published: (2013-01-01)

Correction: Estrogen Signalling and the Metabolic Syndrome: Targeting the Hepatic Estrogen Receptor Alpha Action.
by: Marko Matic, et al.
Published: (2019-01-01)

Estrogen and inflammation modulate estrogen receptor alpha expression in specific tissues of the temporomandibular joint
by: Bellinger Larry L, et al.
Published: (2009-12-01)

Down-regulation of estrogen receptor-alpha and rearranged during transfection tyrosine kinase is associated with withaferin a-induced apoptosis in MCF-7 breast cancer cells
by: Samadi Abbas K, et al.
Published: (2011-10-01)

A Role for Estrogen Receptor alpha36 in Cancer Progression
by: Maria Teresa Pagano, et al.
Published: (2020-07-01)

Whole-genome cartography of estrogen receptor alpha binding sites.
by: Chin-Yo Lin, et al.
Published: (2007-06-01)

Pancreatic insulin content regulation by the estrogen receptor ER alpha.
by: Paloma Alonso-Magdalena, et al.
Published: (2008-04-01)

Ligands specify estrogen receptor alpha nuclear localization and degradation
by: Caze-Subra Stéphanie, et al.
Published: (2010-12-01)

Behavioral Disturbances in Estrogen-Related Receptor alpha-Null Mice
by: Huxing Cui, et al.
Published: (2015-04-01)

Steroid-Functionalized Titanocenes: Docking Studies with Estrogen Receptor Alpha
by: Li Ming Gao, et al.
Published: (2016-11-01)

Estradiol accelerates liver regeneration through estrogen receptor α
by: Tsugawa Y, et al.
Published: (2019-07-01)

The role of estrogen receptors alpha and beta in the development of uterine leiomyomas
by: Koomson, Jacqueline Nyarkoa
Published: (2017)

Targeted Deletion of Estrogen Receptor Alpha in Mouse Pituitary Lactotrophs
by: Minges, Cheryl
Published: (2011)

Estrogen Receptor Alpha in the Medial Preopic Area Mediates Male Rat Sexual Responses to Estrogen
by: Russell, Nancy
Published: (2010)

Estrogen-mediated hemangioma-derived stem cells through estrogen receptor-α for infantile hemangioma
by: Zhang L, et al.
Published: (2017-07-01)

Estrogen-Related Receptor α (ERRα) and G Protein-Coupled Estrogen Receptor (GPER) Synergistically Indicate Poor Prognosis in Patients with Triple-Negative Breast Cancer
by: Ye S, et al.
Published: (2020-09-01)

An in silico study to search for human estrogen receptor-alpha dimerization motif(s)
by: King, Candace
Published: (2015)

Estrogen alpha receptor antagonists for the treatment of breast cancer: a review
by: Deepika Sharma, et al.
Published: (2018-10-01)

Alpha-defensins 1-3 release by dendritic cells is reduced by estrogen
by: Sperling Rhoda, et al.
Published: (2011-08-01)

Gene expression of estrogen receptor-alpha in orbital fibroblasts in Graves’ ophthalmopathy
by: Sarah Santiloni Cury, et al.

Cohesin is required for expression of the estrogen receptor-alpha (<it>ESR1</it>) gene
by: Prenzel Tanja, et al.
Published: (2012-08-01)