Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities

Some hitherto unknown novel bismesoionic compounds, 3-[4/3-(5H/substituted- 2-sulphido-1,3,4-thiadiazolium-4-carbonyl)phenyl]sydnones 5a–d and 6a-d and 4-[4-(5H/substituted-2-sulphido-1,3,4-thiadiazolium)benzoyl]-5H/substituted-1,3,4-thiadiazolium-2-thiolates 9a–d have been synthesized from 3-[(hydr...

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Main Authors: JOHNSON J. JOGUL, BHARATI V. BADAMI
Format: Article
Language:English
Published: Serbian Chemical Society 2006-09-01
Series:Journal of the Serbian Chemical Society
Subjects:
Online Access:http://www.shd.org.yu/HtDocs/SHD/Vol71/No8-9/JSCS_V71_No8-9-01.pdf
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spelling doaj-8701db124c2c42b79b33c5255f1204002020-11-25T00:49:14ZengSerbian Chemical Society Journal of the Serbian Chemical Society0352-51392006-09-01718-9851860Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activitiesJOHNSON J. JOGULBHARATI V. BADAMISome hitherto unknown novel bismesoionic compounds, 3-[4/3-(5H/substituted- 2-sulphido-1,3,4-thiadiazolium-4-carbonyl)phenyl]sydnones 5a–d and 6a-d and 4-[4-(5H/substituted-2-sulphido-1,3,4-thiadiazolium)benzoyl]-5H/substituted-1,3,4-thiadiazolium-2-thiolates 9a–d have been synthesized from 3-[(hydrazinocarbonyl)phenyl] sydnones 1 and 2. Afew of these compounds exhibited in vitro antitubercular activity and also antimicrobial activity higher than the employed reference drugs.http://www.shd.org.yu/HtDocs/SHD/Vol71/No8-9/JSCS_V71_No8-9-01.pdf3-[4/3-(hydrazinocarbonyl)phenyl]sydnonesbismesoionic compounds
collection DOAJ
language English
format Article
sources DOAJ
author JOHNSON J. JOGUL
BHARATI V. BADAMI
spellingShingle JOHNSON J. JOGUL
BHARATI V. BADAMI
Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
Journal of the Serbian Chemical Society
3-[4/3-(hydrazinocarbonyl)phenyl]sydnones
bismesoionic compounds
author_facet JOHNSON J. JOGUL
BHARATI V. BADAMI
author_sort JOHNSON J. JOGUL
title Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
title_short Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
title_full Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
title_fullStr Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
title_full_unstemmed Sydnone derivatives as synthons for novel bismesoionic compounds.Synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
title_sort sydnone derivatives as synthons for novel bismesoionic compounds.synthesis of 3-(2-sulphido-1,3,4-thiadiazolium-4-carbonylphenyl) sydnones and 4-[4-(2-sulphido-1,3,4-thiadiazolium) benzoyl]-1,3,4-thiadiazolium-2-thiolates from 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones, and their antimicrobial and antitubercular activities
publisher Serbian Chemical Society
series Journal of the Serbian Chemical Society
issn 0352-5139
publishDate 2006-09-01
description Some hitherto unknown novel bismesoionic compounds, 3-[4/3-(5H/substituted- 2-sulphido-1,3,4-thiadiazolium-4-carbonyl)phenyl]sydnones 5a–d and 6a-d and 4-[4-(5H/substituted-2-sulphido-1,3,4-thiadiazolium)benzoyl]-5H/substituted-1,3,4-thiadiazolium-2-thiolates 9a–d have been synthesized from 3-[(hydrazinocarbonyl)phenyl] sydnones 1 and 2. Afew of these compounds exhibited in vitro antitubercular activity and also antimicrobial activity higher than the employed reference drugs.
topic 3-[4/3-(hydrazinocarbonyl)phenyl]sydnones
bismesoionic compounds
url http://www.shd.org.yu/HtDocs/SHD/Vol71/No8-9/JSCS_V71_No8-9-01.pdf
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