Bis-Lactam Peptide [<i>i</i>, <i>i</i>+4]-Stapling with α-Methylated Thialysines

Bis-Lactam Peptide [<i>i</i>, <i>i</i>+4]-Stapling with α-Methylated Thialysines

Four bis-lactam [<i>i</i>, <i>i</i>+4]-stapled peptides with <span style="font-variant: small-caps;">d</span>- or <span style="font-variant: small-caps;">l</span>-α-methyl-thialysines were constructed on a model peptide sequence der...

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Bibliographic Details
Main Authors:	Bo Wu, Weiping Zheng
Format:	Article
Language:	English
Published:	MDPI AG 2020-10-01
Series:	Molecules
Subjects:	peptide stapling bis-lactam [<i>i</i>, <i>i</i>+4]-stapling α-methyl-thialysine % α-helicity proteolytic stability
Online Access:	https://www.mdpi.com/1420-3049/25/19/4506

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