Synthesis, Antifungal Activities and Molecular Docking Studies of Benzoxazole and Benzothiazole Derivatives

Synthesis, Antifungal Activities and Molecular Docking Studies of Benzoxazole and Benzothiazole Derivatives

Based on benzoxazole and benzothiazole scaffold as an important pharmacophore, two series of 2-(aryloxymethyl) benzoxazole and benzothiazole derivatives were synthesized and their antifungal effects against eight phytopathogenic fungi were evaluated. Compounds 5a, 5b, 5h, and 5i exhibited significan...

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Bibliographic Details
Main Authors:	Bo Luo, Ding Li, An-Ling Zhang, Jin-Ming Gao
Format:	Article
Language:	English
Published:	MDPI AG 2018-09-01
Series:	Molecules
Subjects:	benzoxazole derivatives benzothiazole derivatives fungicidal activity plant pathogens structure-activity relationships molecular docking
Online Access:	http://www.mdpi.com/1420-3049/23/10/2457

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