Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures

Bibliographic Details
Main Authors: Dirk Lindenblatt, Anna Nickelsen, Violetta M. Applegate, Jennifer Hochscherf, Benedict Witulski, Zouhair Bouaziz, Christelle Marminon, Maria Bretner, Marc Le Borgne, Joachim Jose, Karsten Niefind
Format: Article
Language:English
Published: American Chemical Society 2019-03-01
Series:ACS Omega
Online Access:http://dx.doi.org/10.1021/acsomega.8b03415
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spelling doaj-6c5bcdc4d49e447faba4e5a030c89f662020-11-25T03:33:47ZengAmerican Chemical SocietyACS Omega2470-13432019-03-01435471547810.1021/acsomega.8b03415Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ StructuresDirk Lindenblatt0Anna Nickelsen1Violetta M. Applegate2Jennifer Hochscherf3Benedict Witulski4Zouhair Bouaziz5Christelle Marminon6Maria Bretner7Marc Le Borgne8Joachim Jose9Karsten Niefind10Department für Chemie, Institut für Biochemie, Universität zu Köln, Köln, GermanyInstitut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Münster, GermanyDepartment für Chemie, Institut für Biochemie, Universität zu Köln, Köln, GermanyDepartment für Chemie, Institut für Biochemie, Universität zu Köln, Köln, GermanyDepartment für Chemie, Institut für Biochemie, Universität zu Köln, Köln, GermanyEA 4446 Bioactive Molecules and Medicinal Chemistry, SFR Santé Lyon-Est CNRS UMS 3453 - INSERM US7, Faculté de Pharmacie-ISPB, Université Claude Bernard Lyon 1, Lyon Cedex 8, FranceEA 4446 Bioactive Molecules and Medicinal Chemistry, SFR Santé Lyon-Est CNRS UMS 3453 - INSERM US7, Faculté de Pharmacie-ISPB, Université Claude Bernard Lyon 1, Lyon Cedex 8, FranceFaculty of Chemistry, Warsaw University of Technology, Warsaw, PolandEA 4446 Bioactive Molecules and Medicinal Chemistry, SFR Santé Lyon-Est CNRS UMS 3453 - INSERM US7, Faculté de Pharmacie-ISPB, Université Claude Bernard Lyon 1, Lyon Cedex 8, FranceInstitut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, Münster, GermanyDepartment für Chemie, Institut für Biochemie, Universität zu Köln, Köln, Germanyhttp://dx.doi.org/10.1021/acsomega.8b03415
collection DOAJ
language English
format Article
sources DOAJ
author Dirk Lindenblatt
Anna Nickelsen
Violetta M. Applegate
Jennifer Hochscherf
Benedict Witulski
Zouhair Bouaziz
Christelle Marminon
Maria Bretner
Marc Le Borgne
Joachim Jose
Karsten Niefind
spellingShingle Dirk Lindenblatt
Anna Nickelsen
Violetta M. Applegate
Jennifer Hochscherf
Benedict Witulski
Zouhair Bouaziz
Christelle Marminon
Maria Bretner
Marc Le Borgne
Joachim Jose
Karsten Niefind
Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
ACS Omega
author_facet Dirk Lindenblatt
Anna Nickelsen
Violetta M. Applegate
Jennifer Hochscherf
Benedict Witulski
Zouhair Bouaziz
Christelle Marminon
Maria Bretner
Marc Le Borgne
Joachim Jose
Karsten Niefind
author_sort Dirk Lindenblatt
title Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
title_short Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
title_full Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
title_fullStr Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
title_full_unstemmed Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures
title_sort diacritic binding of an indenoindole inhibitor by ck2α paralogs explored by a reliable path to atomic resolution ck2α′ structures
publisher American Chemical Society
series ACS Omega
issn 2470-1343
publishDate 2019-03-01
url http://dx.doi.org/10.1021/acsomega.8b03415
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