Synthesis and biological evaluation of some novel pyrazole, isoxazole, benzoxazepine, benzothiazepine and benzodiazepine derivatives bearing an aryl sulfonate moiety as antimicrobial and anti-inflammatory agents

Synthesis and biological evaluation of some novel pyrazole, isoxazole, benzoxazepine, benzothiazepine and benzodiazepine derivatives bearing an aryl sulfonate moiety as antimicrobial and anti-inflammatory agents

A new series of pyrazole, isoxazole, benzoxazepine, benzothiazepine and benzodiazepine derivatives were prepared by the multi-component cyclo-condensation reaction of 1-phenyl-3-(2-(tosyloxy)phenyl)propane-1,3-dione, N,N-dimethylformamide dimethyl acetal and hydrazine or hydroxylamine hydrochloride...

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Bibliographic Details
Main Authors:	Babasaheb V. Kendre, Mahadev G. Landge, Sudhakar R. Bhusare
Format:	Article
Language:	English
Published:	Elsevier 2019-12-01
Series:	Arabian Journal of Chemistry
Online Access:	http://www.sciencedirect.com/science/article/pii/S1878535215000258

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