Synthesis and in vitro anti-HIV-1 evaluation of some N-arylsulfonyl-3-formylindoles
As our ongoing work on research of anti-HIV-1 inhibitors, fifteen N-arylsulfonyl-3-formylindoles (3a-o) were designed and prepared through two step synthetic route. Firstly, 3-formylindoles (2a-c) were synthesized via the Vilsmeier-Haack reaction. Subsequently, treatment of 2a-c with the appropriate...
Main Authors: | , , , , |
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Format: | Article |
Language: | English |
Published: |
Universidade de São Paulo
2018-11-01
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Series: | Brazilian Journal of Pharmaceutical Sciences |
Subjects: | |
Online Access: | http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1984-82502018000300605&lng=en&tlng=en |