Microwave Assisted Improved Method for the Synthesis of Pyrazole Containing 2,4,-Disubstituted Oxazole-5-one and their Antimicrobial Activity

Microwave Assisted Improved Method for the Synthesis of Pyrazole Containing 2,4,-Disubstituted Oxazole-5-one and their Antimicrobial Activity

Disubstituted oxazol-5-one and pyrazoles are known to exhibit various biological activities. Therefore, in this work, we designed pyrazole containing 2,4-disubstituted oxazol-5-one (3a-g) as a new class of antimicrobial agents. Synthesis of titled compounds was carried out by two different methods....

Full description

Bibliographic Details
Main Authors:	N. D. Argade, B. K. Kalrale, C. H. Gill
Format:	Article
Language:	English
Published:	Hindawi Limited 2008-01-01
Series:	E-Journal of Chemistry
Online Access:	http://dx.doi.org/10.1155/2008/265131

Similar Items

Synthesis of some 1-aryl-3,5-disubstituted-pyrazoles by N-arylation of 3,5-disubstituted-pyrazoles with 4-fluoro and 2-fluoronitrobenzene under microwave irradiation and classical heating
by: Ibrahim Bouabdallah, et al.
Published: (2006-08-01)

Efficient One-Pot, Two-Component Modular Synthesis of 3,5-Disubstituted Pyrazoles
by: Samy Mohamady, et al.
Published: (2018-11-01)

Synthesis and biological evaluation of newer analogues of 2,5-disubstituted 1,3,4-oxadiazole containing pyrazole moiety as antimicrobial agents
by: Shridhar Malladi, et al.
Published: (2014-12-01)

Synthesis and Cytotoxic Activities of 4,5-Disubstituted isoxazoles and pyrazoles
by: Hon-Cha Huang, et al.
Published: (2009)

Synthesis and antimicrobial activity of pyrazole nucleus containing 2-thioxothiazolidin-4-one derivatives
by: H. B’Bhatt, et al.
Published: (2017-05-01)

Hypervalent Iodine(III) Reagent Promoted Oxidative Cyclization of Propargyl Amides: Facile synthesis of 2,5- Disubstituted Oxazolines and Oxazoles
by: Shih-Chen Lin, et al.
Published: (2014)

Formation of thiadiazole, thiadiazine, thiadiazepine and pyrazole derivatives in the reaction of 2,4-disubstituted thiosemicarbazides with tetracyanoethylene
by: Alaa A. Hassan, et al.
Published: (2018-03-01)

Synthesis of the Oxazole-Containing Natural Products Siphonazole and Telomestatin
by: Linder, Jorg
Published: (2009)

Synthesis and characterization of some heterocyclic including oxazoles,Thiazoles, Pyridazines, phthalizines and Pyrazoles with evaluating of biological activity.
by: Baghdad Science Journal
Published: (2013-09-01)

Synthesis, Characterization and Biological Activity Evaluation of Some Pyrazoles, Thiazoles and Oxazoles Derived from 2-Mercaptoaniline
by: Ahmood Kh. Jebur AL-Joubory, et al.
Published: (2021-03-01)

Novel Ethyl 1,5-Disubstituted-1H-Pyrazole-3-Carboxylates as a New Class of Antimicrobial Agents
by: Radwan Awwad A., et al.
Published: (2014-09-01)

Microwave-assisted synthesis, characterization and biological activity of novel pyrazole derivatives
by: Theivendren Panneer Selvam, et al.
Published: (2014-12-01)

Microwave-assisted multi-component synthesis of 3’-indolyl substituted pyrano[2,3-c]pyrazoles and their antimicrobial activity
by: Kathrotiya Harshad G., et al.
Published: (2012-01-01)

Microwave-assisted synthesis of new pyrazole derivatives bearing 1,2,3-triazole scaffold as potential antimicrobial agents
by: Ashok Dongamanti, et al.
Published: (2017-01-01)

An Efficient One-Pot Catalyzed Synthesis of 2,4-Disubstituted 5-Nitroimidazoles Displaying Antiparasitic and Antibacterial Activities
by: Fanny Mathias, et al.
Published: (2017-08-01)

A microwave-catalyzed rapid, efficient and ecofriendly synthesis of substituted pyrazol-5-ones
by: RAHUL P. GAVANDE, et al.
Published: (2003-10-01)

Microwave-assisted one pot three-component synthesis of some novel pyrazole scaffolds as potent anticancer agents
by: Sobhi M. Gomha, et al.
Published: (2017-05-01)

Naturally Occurring Oxazole-Containing Peptides
by: Jessica T. Mhlongo, et al.
Published: (2020-04-01)

Recent Advances in the Synthesis of Oxazole-Based Molecules via van Leusen Oxazole Synthesis
by: Xunan Zheng, et al.
Published: (2020-03-01)

Simple two-step synthesis of 2,4-disubstituted pyrroles and 3,5-disubstituted pyrrole-2-carbonitriles from enones
by: Murat Kucukdisli, et al.
Published: (2014-02-01)

A facile one-pot synthesis of novel 2,5-disubstituted-1,3,4-oxadiazoles under conventional and microwave conditions and evaluation of their in vitro antimicrobial activities
by: Nida N. Farshori, et al.
Published: (2017-05-01)

Synthesis of 2,4-Disubstituted Pyrimidines of Possible Biological Interest
by: Barnes, Samuel
Published: (2008)

A radical sterocontrolled synthesis of 2,4-disubstituted piperidines
by: Gandon, Lucile Alice
Published: (2003)

Microwave-Assisted Synthesis of Mono- and Disubstituted 4-Hydroxyacetophenone Derivatives via Mannich Reaction: Synthesis, XRD and HS-Analysis
by: Ghadah Aljohani, et al.
Published: (2019-02-01)

Microwave-assisted synthesis of mono- and disubstituted 4-hydroxyacetophenone derivatives via Mannich reaction: synthesis, XRD and HS-analysis
by: Aljohani, Ghadah, et al.
Published: (2019)

Synthesis and research of derived oxazol-5-ones based on α,β – unsaturated ketones
by: Сергей Александрович Петров
Published: (2015-11-01)

Study of Facial and Regio Selectivity on 2,4-Disubstituted Adamantanes and 2,5-Disubstituted Adamantylidenefulvenes
by: Jean- Ho Chu, et al.
Published: (1999)

Synthesis of new trifluoromethyl-containing 1-(3,5-dialkyl-4-hydroxybenzyl)-pyrazole and -pyrazol-5-one deriatives and their corresponding aroxyls
by: Dinoiu Vasile, et al.
Published: (2006-01-01)

Synthesis of new trifluoromethyl-containing 1-(3,5-dialkyl-4-hydroxybenzyl)-pyrazole and -pyrazol-5-one deriatives and their corresponding aroxyls
by: VASILE DINOIU, et al.
Published: (2006-04-01)

Synthesis, characterization and antimicrobial evaluation of 2,5-disubstituted-4-thiazolidinone derivatives
by: Aakash Deep, et al.
Published: (2014-07-01)

Synthesis, antimicrobial and in silico studies of new 2.5-disubstituted benzoxazole derivative
by: Meryem Erol, et al.
Published: (2021-06-01)

Conventional and microwave assisted synthesis of 1,4-disubstituted 1,2,3-triazoles from Huisgen cycloaddition
by: Juan Ignacio Sarmiento-Sanchez, et al.
Published: (2011-05-01)

One-pot microwave-assisted synthesis of 2,5-bis(pyrazol-4-yl)[1,3]thiazolo[5,4-d][1,3]thiazoles from pyrazole-4-carbaldehydes and dithiooxamide
by: Lyubov K. Papernaya, et al.
Published: (2016-09-01)

Microwave-assisted one-pot synthesis of 2-amino-6,7-disubstituted-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-4(3H)-one without catalyst
by: Shujiang Tu, et al.
Published: (2005-06-01)

Room Temperature Copper(II)-Catalyzed Oxidative Cyclization of Enamides to 2,5-Disubstituted Oxazoles via Vinylic C-H Functionalization
by: Cheung, Chi Wai, et al.
Published: (2013)

A microwave-catalyzed rapid, efficient and ecofriendly synthesis of substituted pyrazol-5-ones (Short communication)
by: Dabholkar Vijay V., et al.
Published: (2003-01-01)

Synthesis of 2,4-disubstituted quinazolines promoted by deep eutectic solvent
by: Rajkumar Romeshkumar Singh, et al.
Published: (2021-01-01)

Thiazole and Oxazole Alkaloids: Isolation and Synthesis
by: Gloria Serra, et al.
Published: (2010-11-01)

Microwave-Assisted Traceless Synthesis of Disubstituted Indole Alkaloids, pyrrolo[3,2-c]quinolines and Piperazino-Oxazinones derivatives.
by: Wen-Pin Yeh, et al.
Published: (2008)

Catalyst-and organic solvent-free synthesis, structural, and theoretical studies of 1-arylidenamino-2,4-disubstituted-2-imidazoline-5-ones
by: Wessam Saaed, et al.
Published: (2020-01-01)