C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors

Bibliographic Details
Main Authors: Dharshini Ganeshapillai, L. W. Lawrence Woo, Mark P. Thomas, Atul Purohit, Barry V. L. Potter
Format: Article
Language:English
Published: American Chemical Society 2018-09-01
Series:ACS Omega
Online Access:http://dx.doi.org/10.1021/acsomega.8b01383
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spelling doaj-2e29194f912d47a5a2b1bbe6f389e4802020-11-25T03:32:22ZengAmerican Chemical SocietyACS Omega2470-13432018-09-0139107481077210.1021/acsomega.8b01383C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase InhibitorsDharshini Ganeshapillai0L. W. Lawrence Woo1Mark P. Thomas2Atul Purohit3Barry V. L. Potter4Medicinal Chemistry, Department of Pharmacy and Pharmacology, University of Bath, Bath, U.K.Medicinal Chemistry, Department of Pharmacy and Pharmacology, University of Bath, Bath, U.K.Medicinal Chemistry, Department of Pharmacy and Pharmacology, University of Bath, Bath, U.K.Section of Investigative Medicine, Diabetes, Endocrinology & Metabolism, Imperial College London, London, U.K.Medicinal Chemistry & Drug Discovery, Department of Pharmacology, University of Oxford, Oxford, U.K.http://dx.doi.org/10.1021/acsomega.8b01383
collection DOAJ
language English
format Article
sources DOAJ
author Dharshini Ganeshapillai
L. W. Lawrence Woo
Mark P. Thomas
Atul Purohit
Barry V. L. Potter
spellingShingle Dharshini Ganeshapillai
L. W. Lawrence Woo
Mark P. Thomas
Atul Purohit
Barry V. L. Potter
C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
ACS Omega
author_facet Dharshini Ganeshapillai
L. W. Lawrence Woo
Mark P. Thomas
Atul Purohit
Barry V. L. Potter
author_sort Dharshini Ganeshapillai
title C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
title_short C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
title_full C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
title_fullStr C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
title_full_unstemmed C‑3- and C‑4-Substituted Bicyclic Coumarin Sulfamates as Potent Steroid Sulfatase Inhibitors
title_sort c‑3- and c‑4-substituted bicyclic coumarin sulfamates as potent steroid sulfatase inhibitors
publisher American Chemical Society
series ACS Omega
issn 2470-1343
publishDate 2018-09-01
url http://dx.doi.org/10.1021/acsomega.8b01383
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AT markpthomas c3andc4substitutedbicycliccoumarinsulfamatesaspotentsteroidsulfataseinhibitors
AT atulpurohit c3andc4substitutedbicycliccoumarinsulfamatesaspotentsteroidsulfataseinhibitors
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