The Ring Transformation of 3-Methyl-5-nitropyrimidin-4(3H)-one

The Ring Transformation of 3-Methyl-5-nitropyrimidin-4(3H)-one

3-Methyl-5-nitropyrimidin-4(3H)-one readily reacts with carbonyl compounds to produce three kinds of ring transformations. The nitropyrimidinone behaves as the synthetic equivalent of activated diformylamine affording 3,5-difunctionalized 4-pyridones, 4,5-disubstituted pyrimidines and functionalized...

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Bibliographic Details
Main Authors:	Masahiro Ariga, Yasuo Tohda, Kazushige Hori, Mina Tamura, Nagatoshi Nishiwaki
Format:	Article
Language:	English
Published:	MDPI AG 2003-06-01
Series:	Molecules
Subjects:	Nitropyrimidinone ring transformation pyridone pyrimidine aminopyridine
Online Access:	http://www.mdpi.com/1420-3049/8/6/500/

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